Produktbild: ADME Technologies

ADME Technologies

239,99 €

inkl. gesetzl. MwSt., Versandkostenfrei


Beschreibung

Produktdetails

Einband

Gebundene Ausgabe

Erscheinungsdatum

20.04.2012

Herausgeber

Sekhar Surapaneni + weitere

Verlag

John Wiley & Sons Inc

Seitenzahl

624

Maße (L/B/H)

28,6/22,1/3,8 cm

Gewicht

1803 g

Auflage

1. Auflage

Sprache

Englisch

ISBN

978-0-470-54278-1

Beschreibung

Rezension

"This book fills time needs of ADME researchers and provides a fine reference book for scientists engaged in the areas of medicinal chemistry, pharmaceutics, bioanalytical sciences, pharmacology and toxicology in academia and pharmaceutical industry." (British Toxicology Society, 1 July 2013)

Produktdetails

Einband

Gebundene Ausgabe

Erscheinungsdatum

20.04.2012

Herausgeber

Verlag

John Wiley & Sons Inc

Seitenzahl

624

Maße (L/B/H)

28,6/22,1/3,8 cm

Gewicht

1803 g

Auflage

1. Auflage

Sprache

Englisch

ISBN

978-0-470-54278-1

Herstelleradresse

Libri GmbH
Europaallee 1
36244 Bad Hersfeld
DE

Email: gpsr@libri.de

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  • Produktbild: ADME Technologies
  • FOREWORD xxi
    Lisa A. Shipley
     
    PREFACE xxv
    Donglu Zhang and Sekhar Surapaneni
     
    CONTRIBUTORS xxvii
     
    PART A ADME: OVERVIEW AND CURRENT TOPICS 1
     
    1 Regulatory Drug Disposition and NDA Package Including MIST 3
    Sekhar Surapaneni
     
    References 12
     
    2 Optimal ADME Properties for Clinical Candidate and Investigational New Drug (IND) Package 15
    Rajinder Bhardwaj and Gamini Chandrasena
     
    References 25
     
    3 Drug Transporters in Drug Interactions and Disposition 29
    Imad Hanna and Ryan M. Pelis
     
    References 46
     
    4 Pharmacological and Toxicological Activity of Drug Metabolites 55
    W. Griffith Humphreys
     
    References 63
     
    5 Improving the Pharmaceutical Properties of Biologics in Drug Discovery: Unique Challenges and Enabling Solutions 67
    Jiwen Chen and Ashok Dongre
     
    References 75
     
    6 Clinical Dose Estimation Using Pharmacokinetic/Pharmacodynamic Modeling and Simulation 79
    Lingling Guan
     
    References 93
     
    7 Pharmacogenomics and Individualized Medicine 95
    Anthony Y.H. Lu and Qiang Ma
     
    Disclaimer 105
     
    Contact Information 105
     
    References 105
     
    8 Overview of Drug Metabolism and Pharmacokinetics with Applications in Drug Discovery and Development in China 109
    Chang-Xiao Liu
     
    References 125
     
    PART B ADME SYSTEMS AND METHODS 129
     
    9 Technical Challenges and Recent Advances of Implementing Comprehensive ADMET Tools in Drug Discovery 131
    Jianling Wang and Leslie Bell
     
    Acknowledgments 155
     
    References 155
     
    10 Permeability and Transporter Models in Drug Discovery and Development 161
    Praveen V. Balimane, Yong-Hae Han, and Saeho Chong
     
    References 167
     
    11 Methods for Assessing Blood-Brain Barrier Penetration in Drug Discovery 169
    Li Di and Edward H. Kerns
     
    References 174
     
    12 Techniques for Determining Protein Binding in Drug Discovery and Development 177
    Tom Lloyd
     
    Acknowledgment 185
     
    References 185
     
    13 Reaction Phenotyping 189
    Chun Li and Nataraj Kalyanaraman
     
    References 206
     
    14 Fast and Reliable CYP Inhibition Assays 213
    Ming Yao, Hong Cai, and Mingshe Zhu
     
    References 230
     
    15 Tools and Strategies for the Assessment of Enzyme Induction in Drug Discovery and Development 233
    Adrian J. Fretland, Anshul Gupta, Peijuan Zhu, and Catherine L. Booth-Genthe
     
    References 246
     
    16 Animal Models for Studying Drug Metabolizing Enzymes and Transporters 253
    Kevin L. Salyers and Yang Xu
     
    Acknowledgments 271
     
    References 271
     
    17 Milk Excretion and Placental Transfer Studies 277
    Matthew Hoffmann and Adam Shilling
     
    References 289
     
    18 Human Bile Collection for ADME Studies 291
    Suresh K. Balani, Lisa J. Christopher, and Donglu Zhang
     
    Acknowledgment 297
     
    References 297
     
    PART C ANALYTICAL TECHNOLOGIES 299
     
    19 Current Technology and Limitation of LC-MS 301
    Cornelis E.C.A. Hop
     
    References 314
     
    20 Application of Accurate Mass Spectrometry for Metabolite Identification 317
    Zhoupeng Zhang and Kaushik Mitra
     
    References 329
     
    21 Applications of Accelerator Mass Spectrometry (AMS) 331
    Xiaomin Wang, Voon Ong, and Mark Seymour
     
    References 337
     
    22 Radioactivity Profiling 339
    Wing Wah Lam, Jose Silva, and Heng-Keang Lim
     
    Acknowledgments 349
     
    References 349
     
    23 A Robust Methodology for Rapid Structure Determination of Microgram-Level Drug Metabolites by NMR Spectroscopy 353
    Kim A. Johnson, Stella Huang, and Yue-Zhong Shu
     
    References 362
     
    24 Superc