Medicinal Chemistry is emerged as highly interdisciplinary science, since it facilitates towards activity guided synthesis of drug molecules. This field includes the knowledge from gene therapy and computer aided molecular modeling techniques also. Dr. Bhima Sridevi main author of this amazing book has an upshot of vision to develop one pot efficient synthetic methodologies to attain diversely substituted scaffolds of biological interest. I believe that this book assist the undergraduate and graduate students to comprehend the facile synthetic methodologies that allows for the synthesis of biologically relevant diverse Benzo fused N- heterocycles interestingly. Since all the chapters were clearly explained by including synthetic route along with analogues, Screening results, Docking results, detailed characterization data like 1H NMR,13C NMR, HRMS(ESI) etc.